Tranexamic acid is a well-studied oral medication originally used to reduce bleeding. In recent years, it has gained recognition in dermatology for its ability to fade stubborn hyperpigmentation such as melasma, sunspots and post-inflammatory hyperpigmentation. It works by reducing inflammation and blocking signals that trigger excess melanin production.
Tranexamic acid works by inhibiting the activity of plasmin, which helps reduce inflammation in the skin and interrupts the pathways that lead to melanin overproduction. This makes it especially helpful for treating pigment triggered by sun exposure, hormones or chronic inflammation.
It is often prescribed in low doses as a daily oral supplement and is generally well-tolerated. In some cases, topical or injectable forms may be used, but oral medication remains the most common approach for persistent hyperpigmentation.
While tranexamic acid is specific to hyperpigmentation, other oral medications may be prescribed by doctors for related concerns such as acne or hair loss:
These treatments are only recommended after a full consultation and blood work where necessary. Our doctors will assess whether oral medication is suitable and safe for each individual.
Yes. It is safe and effective across all skin types, including skin tones prone to hyperpigmentation.
Most people begin to notice visible lightening within 8 to 12 weeks of consistent use.
It is generally well-tolerated. Rare side effects may include stomach discomfort or mild headache. It is not suitable for individuals with a history of blood clots and must be prescribed by a doctor.
It depends on your health condition. A full medical assessment is required before starting oral tranexamic acid to ensure it is safe.
Yes. Sun protection is essential. UV exposure can worsen hyperpigmentation, so daily sunscreen use is strongly recommended.